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TC-S 7005
CAS No. 1082739-92-1
TC-S 7005 ( —— )
产品货号. M26838 CAS No. 1082739-92-1
TC-S 7005 is an inhibitor of Polo-like kinases (IC50s: 4 nM, 24 nM and 214 nM for Plk2, Plk3, and Plk1, respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥1426 | 有现货 |
|
| 5MG | ￥2406 | 有现货 |
|
| 10MG | ￥3588 | 有现货 |
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| 25MG | ￥5816 | 有现货 |
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| 50MG | ￥7995 | 有现货 |
|
| 100MG | ￥10773 | 有现货 |
|
| 500MG | ￥21627 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称TC-S 7005
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述TC-S 7005 is an inhibitor of Polo-like kinases (IC50s: 4 nM, 24 nM and 214 nM for Plk2, Plk3, and Plk1, respectively).
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产品描述TC-S 7005 is an inhibitor of Polo-like kinases (IC50s: 4 nM, 24 nM and 214 nM for Plk2, Plk3, and Plk1, respectively).(In Vitro):In human SR fibroblasts, TC-S 7005(1 μM) obviously causess myofibroblast differentiation and decrease fibroblast proliferation rates .
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同义词——
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通路Cell Cycle/DNA Damage
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靶点PLK
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受体CBP/p300; Cereblon
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研究领域——
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适应症——
化学信息
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CAS Number1082739-92-1
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分子量359.4
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分子式C21H17N3O3
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纯度>98% (HPLC)
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溶解度——
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SMILESC[C@H](Nc1cc2c(noc2cn1)-c1ccc2OCOc2c1)c1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Raghu Vannam, et al. Targeted degradation of the enhancer lysine acetyltransferases CBP and p300. Cell Chem Biol. 2020 Dec 31;S2451-9456(20)30513-4.
产品手册
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